Ketanserin Tartrate is a potent and selective 5HT2A antagonist. It has demonstrated neurogenic, addiction cessation, sleep enhancement, anxiolytic, and anti=psychotic properties, among others
Research Indications: Serotonergic research, Anxiolytic Research, Psychoneurodysfunctional Research, HPPD-related Research.
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Ketanserin is a high-affinity antagonist of the 5-HT2A receptor (Ki = 2-3 nM). However, it also blocks the H1 receptor with high affinity (Ki = 2 nM). In addition, ketanserin less potently antagonizes the α1-adrenergic (Ki = ~40 nM), α2-adrenergic = ~200 nM), 5-HT1D (Ki = ? nM), 5-HT2B (Ki = ? nM),5-HT2C (Ki = 100 nM),5-HT6 (Ki = ~300 nM),5-HT7 (Ki = ? nM),D1 (~300 nM), and D2 (Ki = ~500 nM) receptors. It also blocks the vesicular monoamine transporter (VMAT).
Article on Potential Benefits and Related Pharmacology of Ketanserin
USAGE: For Research Use Only! Not For Use in Humans.